马来酸桂哌齐特,Cinepazide maleate;≥98% (HPLC)

别名:(E)-1- [4-(2-氧代-2-吡咯烷-1-基乙基)哌嗪-1-基] -3-(3,4,5-三甲氧基苯基)丙-2-烯-1-马来酸酯;1-(吡咯烷基-1-羰基)-甲基-4-(3,4,5-三甲氧基肉桂酰基)-哌嗪-马来酸酯;(E)-1-[4-(2-Oxo-2-pyrrolidin-1-ylethyl)piperazin-1-yl]-3-(3,4,5-trimethoxyphenyl)prop-2-en-1-one maleate, 1-(Pyrrolidinyl-1-carbonyl)-methyl-4-(3,4,5-trimethoxycinnamoyl)-piperazine-maleate

Empirical Formula (Hill Notation): C22H31N3O5 · C4H4O4 CAS号: 26328-04-1 分子量: 533.57 MDL编号: MFCD01320526 PubChem化学物质编号: 329825922
制造商品牌: 西格玛 Sigma-Aldrich
货号(SKU): SML1498
CAS号: 26328-04-1
MDL号: MFCD01320526
签订合同 √ 正规发票 √ 技术支持 √ 质量保障 √ 全程可追溯 √
¥1,534.70

说明

一般描述

Cinepazide maleate can be synthesized from ethyl chlorocarbonate activation and (E) 3,4,5-trimethoxycinnamylic acid.[1]
 

生化/生理作用

Cinepazide maleate is a vasodilator used clinically in China used in China for the treatment of cardiovascular and cerebrovascular diseases, and peripheral vascular diseases. Cinepazide maleate is thought to act as a potentiator of adenosine A2 receptors and has also been characterized as a calcium channel blocker. It was withdrawn for agranulocytosis in several countries.
 
 

属性

质量水平

检测方案

≥98% (HPLC)

形式

powder

储存条件

desiccated

颜色

white to beige

溶解性

H2O: 20 mg/mL, clear

储存温度

2-8°C

SMILES string

O=C(O)/C=C\C(O)=O.O=C(N1CCN(CC(N2CCCC2)=O)CC1)/C=C/C3=CC(OC)=C(OC)C(OC)=C3

InChI

1S/C22H31N3O5.C4H4O4/c1-28-18-14-17(15-19(29-2)22(18)30-3)6-7-20(26)25-12-10-23(11-13-25)16-21(27)24-8-4-5-9-24;5-3(6)1-2-4(7)8/h6-7,14-15H,4-5,8-13,16H2,1-3H3;1-2H,(H,5,6)(H,7,8)/b7-6+;2-1-

InChI key

XSTJTOKYCAJVMJ-GVTSEVKNSA-N

 

安全信息

象形图

Exclamation mark

警示用语:

Warning

危险声明

危险分类

Acute Tox. 4 Oral

储存分类代码

11 - Combustible Solids

WGK

WGK 3

商品规格
属性名称属性值
储存温度 Storage temp.2-8°C冷藏
全球实时库存 Availability √美国St. Louis ≥ 20 | 欧洲Eur. ≥ 16 | 東京Tokyo ≥ 5 | 香港与北京 ≥ 20